平安! 发表于 2011-11-9 19:57 . X0 ]2 u1 U. L) s: W
Pazopanib (100 mg/kg/day free base equivalent)
/ s: @: R; H) w, e. [) R3 Z; K 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
, {# J# \2 H) u: l搜索了一下,原料一大堆。5 o4 B3 b; b$ [ \0 b( G: Y# J
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对不起!100mg/kg是用于移植瘤的,我弄错了。
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以下是正版说明书的推荐用量。7 i0 A/ M# W, ~- K5 A
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--------------------- DOSAGE AND ADMINISTRATION ----------------
0 J' r1 n& `9 o6 n( W" q' I* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
2 p, y4 p3 y$ T* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
2 G$ y/ u; E, m, P% c' ]* O---------------------DOSAGE FORMS AND STRENGTHS --------------
! m2 F. D- g! }( D1 v200 mg tablets. (3)
% u$ H3 i6 y- e, y5 m8 n! `% j-------------------------------CONTRAINDICATIONS------------------------ |